2018 Publications

278
Enzymatic fluorination of biotin and tetrazine bioconjugates for pre-targeting approaches to PET imaging.
Phillip T. Lowe, Sergio Dall’Angelo, Andrew Devine, Matteo Zanda, David O’Hagan

ChemBioChem, 2018, 19, 1969-1978
10.1002/cbic.201800234


277
Fluorinated cyclopropanes: synthesis and chemistry of the aryl α,β,β-trifluorocyclopropane motif
Connor J. Thomson, Qingzhi Zhang, Nawaf Al-Maharik, Michael Buehl, David B. Cordes, Alexandra M. Z. Slawin and David O’Hagan

Chem. Commun., 2018, 54, 8415-8418.
10.1039/C8CC04964E


276
Benzylic Functionalisation of Phenyl all‐cis‐2,3,5,6‐Tetrafluorocyclohexane Provides Access to New Organofluorine Building Blocks
Tetiana Bykova, Nawaf Al-Maharik, Alexandra M. Z. Slawin, Michael Bühl, Tomas Lebl, David O’ Hagan.

Chem., Eur. J., 2018, 24, 13290-13296
10.1002/chem.201802166


275
An enzymatic method for C-18F bond formation for PET
David O’Hagan

J. Label. Compd.. Radiopharm., 2018, 61, 461-462
10.1002/jlcr.3523


274
Molecular mechanism of activation of human musk receptors OR5AN1 and OR1A1 by (R)-muscone and diverse other musk-smelling compounds

Lucky Ahmed, Yuetian Zhang, Eric Block, Michael Buehl, Michael J. Corr, Rodrigo A. Cormanich, Sivaji Gundala, Hiroaki Matsunami, David O’Hagan, Mehmet Ozbil, Yi Pan, Sivakumar Sekharan, Nicholas Ten, Mingan Wang, Mingyan Yang, Qingzhi Zhang, Ruina Zhang, Victor S. Batista and Hanyi Zhuang

‎Proc. Natl. Acad. Sci. U.S.A., 2018, 17, E3950-E3958
10.1073/pnas.1713026115


273
Metabolism and hydrophilicity of the polarised ‘Janus face’ all-cis tetrafluorocyclohexyl ring, a candidate motif for drug discovery


272
Synthesis of aryl α,α-difluoroethyl thioethers a novel structure motif in organic chemistry, and extending to aryl α,α-difluoro oxyethers
Ren Tomita, Nawaf Al-Maharik, Andrea Rodil Garcia, Michael Bühl and David O’Hagan

Org. Biomol. Chem., 2018, 16, 1113–1117.
10.1039/c7ob02987j


271
Stereochemical outcomes of C-F activation reactions of benzyl fluoride
Neil S. Keddie, Pier Alexandre Champagne, Justine Desroches, Jean-François Paquin and David O’Hagan

Beilstein J. Org. Chem., 2018, 14, 106–113.
10.3762/bjoc.14.6